SCHEMBL7489376

SCHEMBL7489376

COc1cccc(CN2CCCCC2C(=O)O)c1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
CD274 Q9NZQ7 8/20 0.63
SMN1; SMN2 Q16637 2/20 0.60
POLB P06746 1/20 0.59
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 4/20 0.55
SIGMAR1 Q99720 1/20 0.51
MAPT P10636 1/20 0.51
SPHK1 Q9NYA1 1/20 0.51
PDCD1 Q15116 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30072188 0.86 KMT2A (0.55) MEN1KMT2ACD274POLBKDM4E
SCHEMBL7484491 0.86 MEN1 (0.80) MEN1KMT2ACD274SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL7616379 0.84 SMN1; SMN2 (0.60) CD274SMN1; SMN2KDM4EALDH1A1SIGMAR1
SCHEMBL3563038 0.83 SMN1; SMN2 (0.53) MEN1KMT2ACD274SMN1; SMN2POLB
SCHEMBL3713831 0.81 SMN1; SMN2 (0.63) MEN1KMT2ACD274SMN1; SMN2SPHK1
SCHEMBL16714062 0.81 SMN1; SMN2 (0.63) MEN1KMT2ACD274SMN1; SMN2SPHK1
SCHEMBL3713829 0.81 SMN1; SMN2 (0.63) MEN1KMT2ACD274SMN1; SMN2SPHK1
SCHEMBL7814221 0.81 NPBWR1 (0.58) MEN1KMT2ACD274SMN1; SMN2KDM4E
SCHEMBL7814225 0.81 NPBWR1 (0.58) MEN1KMT2ACD274SMN1; SMN2KDM4E
SCHEMBL21409037 0.81 SMN1; SMN2 (0.56) CD274SMN1; SMN2KDM4ESIGMAR1SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1095839-C 4,5-diaryl oxazole derivatives FUJISAWA PHARMACETICAL CO LTD (JP) 2002-12-11 CN disclosed
EP-0842161-B1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2002-09-18 EP disclosed
EP-1213285-A2 4,5-dipheny-oxazole derivatives and their use as platelet aggregation inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-06-12 EP disclosed
US-6300344-B1 FOR THERAPEUTIC AND/OR PROPHYLACTIC TREATMENT OF ARTERIAL OBSTRUCTION, CEREBROVASCULAR DISEASE, HEPATIC CIRRHOSIS, ARTERIOSCLEROSIS, ISCHEMIC HEART DISEASE, RESTENOSIS AFTER PERCUTANEOUS TRANSLUMINAL CORONARY ANGIOPLASTY, HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-09 US disclosed
US-5972965-A USEFUL FOR INHIBITION OF PLATELET AGGREGATION, VASODILATION, ANTIHYPERTENSIVE ACTIVITY AND PROSTAGLANDIN AGONIST FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-26 US disclosed
CN-1196726-A 4,5-diaryl oxazole derivatives FUJISAWA PHARMACEUTICAL CO (JP) 1998-10-21 CN disclosed
EP-0842161-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-05-20 EP disclosed
WO-1997003973-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-06 WO disclosed