SCHEMBL7490994

SCHEMBL7490994

COc1cc(O)c(CNC(=O)OCCc2ccc(N)cc2)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 9/20 0.48
PTPN1 P18031 2/20 0.45
CYP19A1 P11511 3/20 0.42
CA12 O43570 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
HTR7 P34969 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
NOS2 P35228 1/20 0.42
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CALM1 P0DP23 1/20 0.40
ALOX5 P09917 1/20 0.40
OR51E2 Q9H255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27449774 0.76 PTPN1 (0.56) PTPN1MAPTSMN1; SMN2
SCHEMBL27568244 0.73 PTPN1 (0.47) PTPN1NOS2MAPTSMN1; SMN2
SCHEMBL6598928 0.72 CALM1 (0.44) METPTPN1CYP19A1NOS2CALM1
SCHEMBL3011168 0.70 PPID (0.50) SMN1; SMN2
SCHEMBL22403769 0.70 GLA (0.51) METCA12CA9NPC1RAB9A
SCHEMBL5384679 0.69 CALM1 (0.42) METPTPN1CYP19A1NOS2CALM1
SCHEMBL15650646 0.68 NPC1 (0.51) METNPC1RAB9ASMN1; SMN2NFKB1
SCHEMBL6896587 0.68 NFKB1 (0.58) CYP19A1MAPTALOX5OR51E2NFKB1
SCHEMBL10412135 0.67 CYP19A1 (0.74) PTPN1CYP19A1NOS2ALOX5OR51E2
SCHEMBL5383983 0.66 CDC25C (0.60) CA12CA4CA9MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265891-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2002-12-18 EP disclosed
WO-2001068643-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2001-09-20 WO disclosed