SCHEMBL7493230

SCHEMBL7493230

CCSC(=O)/C(C#N)=C(/C)Nc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.53
HDAC1 Q13547 4/20 0.53
HDAC2 Q92769 4/20 0.53
HDAC8 Q9BY41 4/20 0.53
MAPK10 P53779 2/20 0.46
TP53 P04637 1/20 0.46
DHODH Q02127 1/20 0.46
TSHR P16473 1/20 0.45
KCNH2 Q12809 1/20 0.45
RAB9A P51151 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
HDAC4 P56524 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493234 1.00 HDAC3 (0.53) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7493821 0.84 HDAC3 (0.61) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7493816 0.84 HDAC3 (0.61) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7496099 0.81 ALDH1A1 (0.56) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7496095 0.81 ALDH1A1 (0.56) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL11801755 0.77 MAPT (0.49) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7488992 0.77 MAPT (0.49) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7493927 0.75 MCL1 (0.32) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL7493932 0.75 MCL1 (0.32) HDAC3HDAC1HDAC2HDAC8MAPK10
SCHEMBL4118521 0.74 HDAC8 (0.41) HDAC3HDAC1HDAC2HDAC8TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760362-B1 DIAMINOMETHYLIDENE DERIVATIVE NISSHIN SEIFUN GROUP INC (JP) 2002-08-14 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed