SCHEMBL7493533

SCHEMBL7493533

CC(=C(NC(=O)OCc1ccccc1)C(=O)O)c1ccc(-n2cncn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
HSP90AA1 P07900 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SMYD3 Q9H7B4 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGER1 P34995 1/20 0.38
POLB P06746 1/20 0.38
ROCK1 Q13464 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362764 0.76 MAPT (0.53) MAPTHSP90AA1HTTSMN1; SMN2L3MBTL1
SCHEMBL7362760 0.76 MAPT (0.53) MAPTHSP90AA1HTTSMN1; SMN2L3MBTL1
SCHEMBL8646296 0.74 RAB9A (0.42) MAPTHSP90AA1HTTSMN1; SMN2SMYD3
SCHEMBL5893116 0.71 RAB9A (0.44) MAPTHTTSMN1; SMN2TDP1L3MBTL1
SCHEMBL3050407 0.71 MRGPRX4 (0.43) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL3050406 0.71 MRGPRX4 (0.43) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL4390326 0.69 POLB (0.47) TDP1POLBALDH1A1NPC1RAB9A
SCHEMBL13686645 0.68 MAPT (0.49) MAPTHSP90AA1HTTSMN1; SMN2PTGER1
SCHEMBL8507600 0.68 RAB9A (0.68) MAPTSMN1; SMN2SMYD3NPC1RAB9A
SCHEMBL4667925 0.67 RAB9A (0.62) MAPTSMN1; SMN2L3MBTL1PTGER1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997011960-A1 ANTAGONISTS OF ENDOTHELIN RECEPTORS JAPAT LTD. (CH) 1997-04-03 WO disclosed