SCHEMBL7495240

SCHEMBL7495240

CC(C)(F)c1cc(C(C)(C)F)c2c(c1)C1(CCCNC1)C(=O)N2

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.35
HTR2A P28223 1/20 0.33
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493750 1.00 BACE1 (0.35) BACE1HTR2ACYP3A4CYP2D6CYP2C9
SCHEMBL7504206 0.79 BACE1 (0.47) BACE1HTR2A
SCHEMBL7499439 0.79 BACE1 (0.47) BACE1HTR2A
SCHEMBL7493171 0.79 BACE1 (0.47) BACE1HTR2A
Hydrochloric Acid SCHEMBL7497244 0.78 BACE1 (0.46) BACE1HTR2A
SCHEMBL6640348 0.71 PGR (0.40) BACE1HTR2A
SCHEMBL7500428 0.71 BACE1 (0.49) BACE1HTR2A
SCHEMBL7501462 0.68 BACE1 (0.49) BACE1HTR2ACYP2C9CYP2C19
Acetic Acid SCHEMBL6634718 0.68 PGR (0.38) BACE1HTR2A
SCHEMBL6637300 0.66 PDE7A (0.49) BACE1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202994-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-05-08 EP claimed
WO-2001005790-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2001-01-25 WO claimed
EP-1202994-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-05-08 EP disclosed
WO-2001005790-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2001-01-25 WO disclosed