SCHEMBL7495952

SCHEMBL7495952

COc1c(Cl)cccc1NC(N)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.52
TAS1R3 Q7RTX0 2/20 0.50
TAS1R1 Q7RTX1 2/20 0.50
TAS1R2 Q8TE23 2/20 0.50
CYP1A2 P05177 1/20 0.50
LMNA P02545 3/20 0.48
PDE4D Q08499 1/20 0.48
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 5/20 0.46
GAA P10253 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 2/20 0.44
TOP1 P11387 1/20 0.44
NPC1 O15118 1/20 0.43
CASP3 P42574 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2088326 0.85 RAF1 (0.53) RAF1TAS1R3TAS1R1TAS1R2LMNA
SCHEMBL2088329 0.85 RAF1 (0.53) RAF1TAS1R3TAS1R1TAS1R2CYP1A2
SCHEMBL2093882 0.85 RAF1 (0.53) RAF1TAS1R3TAS1R1TAS1R2LMNA
SCHEMBL2013991 0.83 KMT2A (0.62) RAF1TAS1R3TAS1R1TAS1R2LMNA
SCHEMBL14053368 0.83 RAF1 (0.46) RAF1TAS1R3TAS1R1TAS1R2CYP1A2
SCHEMBL881514 0.83 RAF1 (0.49) RAF1TAS1R3TAS1R1TAS1R2LMNA
SCHEMBL2093879 0.82 RAF1 (0.51) RAF1TAS1R3TAS1R1TAS1R2LMNA
SCHEMBL8493065 0.81 ALDH1A1 (0.59) LMNAALDH1A1KDM4EGAAKMT2A
SCHEMBL7759446 0.80 TAS1R3 (0.50) TAS1R3TAS1R1TAS1R2ALDH1A1KDM4E
SCHEMBL7603112 0.80 KMT2A (0.54) RAF1TAS1R3TAS1R1TAS1R2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0896531-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-10-30 EP disclosed
EP-0896531-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-17 EP disclosed
WO-1997029743-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-21 WO disclosed