SCHEMBL7497779

SCHEMBL7497779

O=COC1(CNS(=O)(=O)c2ccccc2)CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
GBA1 P04062 2/20 0.42
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KEAP1 Q14145 1/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 2/20 0.40
GAA P10253 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSK P43235 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5674483 0.78 GAA (0.42) ALDH1A1LMNASMN1; SMN2KEAP1KDM4E
SCHEMBL5675309 0.75 GAA (0.42) ALDH1A1GBA1LMNAKEAP1KDM4E
SCHEMBL7497785 0.74 BRD4 (0.46) ALDH1A1GBA1LMNASMN1; SMN2KEAP1
SCHEMBL10084139 0.73 SLC6A4 (0.54) ALDH1A1GBA1LMNASMN1; SMN2KEAP1
SCHEMBL9140049 0.71 KEAP1 (0.51) ALDH1A1GBA1LMNASMN1; SMN2KEAP1
SCHEMBL6632034 0.68 CTSK (0.49) ALDH1A1LMNACTSLCTSBCTSK
SCHEMBL6008587 0.68 ALDH1A1 (0.53) ALDH1A1GBA1LMNASMN1; SMN2KEAP1
SCHEMBL6007599 0.66 ALDH1A1 (0.69) ALDH1A1LMNASMN1; SMN2KEAP1KDM4E
SCHEMBL6006902 0.66 ALDH1A1 (0.57) ALDH1A1GBA1LMNASMN1; SMN2KEAP1
SCHEMBL3934921 0.66 ALDH1A1 (0.57) ALDH1A1GBA1LMNASMN1; SMN2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177172-A1 3a,4,5,9b-TETRAHYDRO-1H-BENZ e]INDOL-2-YL AMINE-DERIVED NEUROPEPTIDE Y RECEPTORS LIGANDS USEFUL IN THE TREATMENT OF OBESITY AND OTHER DISORDERS Ortho-McNeil Pharmaceutical, Inc. (US) 2002-02-06 EP disclosed
WO-2000068197-A1 3a,4,5,9b-TETRAHYDRO-1H-BENZ[e]INDOL-2-YL AMINE-DERIVED NEUROPEPTIDE Y RECEPTORS LIGANDS USEFUL IN THE TREATMENT OF OBESITY AND OTHER DISORDERS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-11-16 WO disclosed