SCHEMBL7498016

SCHEMBL7498016

O=C1Nc2ccc([N+](=O)[O-])cc2N=C2CCCC12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
MAPT P10636 3/20 0.46
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
ALDH1A1 P00352 4/20 0.40
GAA P10253 2/20 0.40
CAPN9 O14815 1/20 0.39
CASP3 P42574 1/20 0.39
LMNA P02545 2/20 0.39
RIPK1 Q13546 1/20 0.39
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
PGR P06401 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
POLB P06746 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499602 0.77 MAPT (0.44) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL7502383 0.73 ALDH1A1 (0.43) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL7495533 0.73 GRM2 (0.40) MEN1KMT2AMAPTNOS3NOS1
SCHEMBL17027697 0.69 MAPT (0.64) MEN1KMT2AMAPTALDH1A1CAPN9
SCHEMBL31730190 0.68 CRBN (0.51) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL2717518 0.68 CYP3A4 (0.50) MEN1KMT2AMAPTNOS1CAPN9
SCHEMBL31730207 0.68 ALDH1A1 (0.51) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL6641968 0.67 NOS3 (0.51) MEN1KMT2ANOS3NOS1NOS2
SCHEMBL31748048 0.67 SMN1; SMN2 (0.55) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL7794446 0.66 SIRT2 (0.53) MEN1KMT2AALDH1A1GAACAPN9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed