SCHEMBL7502383

SCHEMBL7502383

O=C1Nc2ccccc2N=C2CCCCC12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
MAPT P10636 8/20 0.43
KMT2A Q03164 4/20 0.43
KDM4E B2RXH2 4/20 0.43
MEN1 O00255 3/20 0.43
LMNA P02545 3/20 0.43
DDB1 Q16531 5/20 0.40
CRBN Q96SW2 5/20 0.40
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
GAA P10253 2/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499602 0.95 MAPT (0.44) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL7495533 0.76 GRM2 (0.40) ALDH1A1MAPTKMT2AKDM4EMEN1
SCHEMBL3880710 0.74 CYP19A1 (0.44) ALDH1A1MAPTKDM4ELMNASMN1; SMN2
SCHEMBL7499826 0.73 NPC1 (0.46) ALDH1A1MAPTDDB1CRBNNPC1
SCHEMBL7498016 0.73 MEN1 (0.46) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL145755 0.73 NOS1 (0.50) ALDH1A1KMT2AKDM4EMEN1
SCHEMBL30074503 0.73 NOS1 (0.50) ALDH1A1KMT2AKDM4EMEN1
SCHEMBL13867519 0.68 NOS1 (0.32) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL9559207 0.67 NOS1 (0.47) ALDH1A1KMT2AMEN1
SCHEMBL7503685 0.64 ALDH1A1 (0.48) ALDH1A1MAPTKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed