SCHEMBL7499085

SCHEMBL7499085

CSc1cc(-c2ccccc2)c(N)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.44
ALDH1A1 P00352 8/20 0.39
GAA P10253 4/20 0.39
LMNA P02545 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDO2 P48775 1/20 0.39
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMARCA2 P51531 1/20 0.35
SMARCA4 P51532 1/20 0.35
PBRM1 Q86U86 1/20 0.35
MEN1 O00255 3/20 0.35
HPGD P15428 3/20 0.35
KMT2A Q03164 3/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27562270 0.84 MAOA (0.41) ALDH1A1GAASMN1; SMN2HSD17B10POLB
SCHEMBL543968 0.75 TDO2 (0.42) ALDH1A1GAALMNASMN1; SMN2TDO2
SCHEMBL5153317 0.74 TDO2 (0.45) ALDH1A1GAALMNATDO2HSD17B10
SCHEMBL544902 0.71 TDO2 (0.42) ALDH1A1GAALMNASMN1; SMN2TDO2
SCHEMBL29139906 0.71 TDO2 (0.42) ALDH1A1GAALMNATDO2HSD17B10
SCHEMBL29272569 0.71 BACE1 (0.48) ALDH1A1GAALMNATDO2HSD17B10
SCHEMBL8069927 0.70 TDO2 (0.39) ALDH1A1GAALMNATDO2HSD17B10
SCHEMBL544129 0.70 TDO2 (0.39) PLAUALDH1A1GAALMNASMN1; SMN2
SCHEMBL10167108 0.70 TDO2 (0.39) PLAUALDH1A1GAALMNATDO2
SCHEMBL15392129 0.70 TDO2 (0.39) PLAUALDH1A1GAALMNATDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171443-A1 BICYCLIC HETEROAROMATIC COMPOUNDS USEFUL AS LH AGONISTS Akzo Nobel N.V. (NL) 2002-01-16 EP disclosed
WO-2000061586-A1 BICYCLIC HETEROAROMATIC COMPOUNDS USEFUL AS LH AGONISTS AKZO NOBEL N.V. (NL) 2000-10-19 WO disclosed