SCHEMBL29139906

SCHEMBL29139906

Nc1sc(Br)cc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.42
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPK1 P28482 2/20 0.41
SMARCA2 P51531 1/20 0.38
SMARCA4 P51532 1/20 0.38
PBRM1 Q86U86 1/20 0.38
BACE1 P56817 1/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
IKBKB O14920 1/20 0.37
MAOA P21397 1/20 0.35
ADORA1 P30542 1/20 0.35
CYP3A4 P08684 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2039997 0.78 ALDH1A1 (0.44) ALDH1A1HSD17B10MAPK1BACE1HPGD
SCHEMBL5153317 0.78 TDO2 (0.45) TDO2ALDH1A1HSD17B10SMARCA2SMARCA4
SCHEMBL22299320 0.77 PTGS1 (0.49) ALDH1A1HSD17B10MAPK1BACE1HPGD
SCHEMBL544902 0.75 TDO2 (0.42) TDO2ALDH1A1HSD17B10SMARCA2SMARCA4
SCHEMBL29272569 0.75 BACE1 (0.48) TDO2ALDH1A1HSD17B10SMARCA2SMARCA4
SCHEMBL543968 0.75 TDO2 (0.42) TDO2ALDH1A1HSD17B10SMARCA2SMARCA4
SCHEMBL2777753 0.75 PTGS2 (0.51) ALDH1A1HSD17B10MAPK1BACE1HPGD
SCHEMBL8069927 0.71 TDO2 (0.39) TDO2ALDH1A1HSD17B10MAPK1SMARCA2
SCHEMBL15392129 0.71 TDO2 (0.39) TDO2ALDH1A1HSD17B10MAPK1SMARCA2
SCHEMBL7499085 0.71 PLAU (0.44) TDO2ALDH1A1HSD17B10MAPK1SMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116897155-A Benzothiazolyl bicyclo [1.1.1] pentane derivatives for the treatment and prevention of hepatitis b virus infection 豪夫迈·罗氏有限公司 2023-10-17 CN disclosed