SCHEMBL7499225

SCHEMBL7499225

O=C(OCc1ccccc1)N(Cc1cccc([N+](=O)[O-])c1)C1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.46
LMNA P02545 3/20 0.45
ALDH1A1 P00352 2/20 0.45
RAB9A P51151 1/20 0.44
HTR2A P28223 1/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
ATM Q13315 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
DCUN1D1 Q96GG9 2/20 0.43
TACR1 P25103 2/20 0.43
UBE2M P61081 1/20 0.43
KCNH2 Q12809 1/20 0.43
POLB P06746 1/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202628 0.84 HTR2A (0.51) HTR2ASLC6A2SLC6A4SLC6A3CYP2D6
Hydrochloric Acid SCHEMBL7138456 0.83 PYCR1 (0.45) PDE1CLMNAALDH1A1RAB9APOLB
SCHEMBL1205029 0.79 CCR5 (0.50) ATMCCR5
SCHEMBL2791615 0.78 HTR2A (0.51) HTR2ASLC6A2SLC6A4SLC6A3CYP2D6
Trifluoroacetic Acid SCHEMBL22588019 0.78 DCUN1D1 (0.53) HTR2ASLC6A2SLC6A4SLC6A3CYP2D6
Hydrochloric Acid SCHEMBL2791610 0.78 HTR2A (0.50) HTR2ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL13543078 0.78 CCR5 (0.46) HTR2ACCR5
SCHEMBL2569626 0.77 CYP1A2 (0.55) PDE1CLMNAALDH1A1RAB9AATM
SCHEMBL803880 0.77 CCR5 (0.54) HTR2ASLC6A2SLC6A4SLC6A3CYP2D6
Hydrochloric Acid SCHEMBL7665198 0.76 CCR5 (0.43) HTR2ACCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265891-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2002-12-18 EP disclosed
WO-2001068643-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2001-09-20 WO disclosed