SCHEMBL7499540

SCHEMBL7499540

COc1cccc(O)c1C(=O)/C=C/c1ncc[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.56
CYP3A4 P08684 2/20 0.53
MAOB P27338 5/20 0.50
MAOA P21397 4/20 0.50
ABCG2 Q9UNQ0 2/20 0.47
CYP1A1 P04798 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
NFKB1 P19838 3/20 0.44
NFKB2 Q00653 3/20 0.44
RELA Q04206 3/20 0.44
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
NR1H4 Q96RI1 1/20 0.43
MEN1 O00255 1/20 0.43
KCNA3 P22001 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
AR P10275 1/20 0.42
TP53 P04637 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499548 1.00 AURKA (0.56) AURKACYP3A4MAOBMAOAABCG2
SCHEMBL7501096 0.92 CYP1A2 (0.48) AURKACYP3A4MAOBMAOAABCG2
SCHEMBL7501089 0.92 CYP1A2 (0.48) AURKACYP3A4MAOBMAOAABCG2
SCHEMBL7501712 0.81 ABCG2 (0.59) CYP3A4MAOBABCG2CYP1A1CYP1A2
SCHEMBL7501717 0.81 ABCG2 (0.59) CYP3A4MAOBABCG2CYP1A1CYP1A2
SCHEMBL20518106 0.78 ABCG2 (0.57) ABCG2
SCHEMBL19880069 0.77 AURKA (0.82) AURKACYP3A4MAOBMAOAABCG2
SCHEMBL20518159 0.75 ABCG2 (0.60) CYP3A4ABCG2CYP1A1CYP1A2CYP2D6
SCHEMBL25193904 0.75 MAPT (0.71) AURKACYP3A4MAOBMAOAABCG2
SCHEMBL7502155 0.75 HSP90AA1 (0.60) CYP3A4MAOBMAOAABCG2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0924202-B1 Imidazole derivative and medicine comprising the same as active ingredient SSP CO LTD (JP) 2002-05-29 EP disclosed
US-6071943-A IMMUNOMODULATORS WHICH SUPPRESS SPECIFIC CYTOKINES, FOR AUTOIMMUNE DISEASES SSP CO. LTD. (JP) 2000-06-06 US disclosed
EP-0924202-A1 Imidazole derivative and medicine comprising the same as active ingredient SSP Co., Ltd. (JP) 1999-06-23 EP disclosed