SCHEMBL7501231

SCHEMBL7501231

O=C1c2ccccc2C(=O)N1CC(=O)N1c2ccccc2N(Cc2ccc(O)cc2)C(=O)[C@H]2CCC[C@H]21

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MT-CO2 P00403 1/20 0.39
ALOX5 P09917 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507674 0.94 ALDH1A1 (0.49) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7507666 0.94 ALDH1A1 (0.49) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7498715 0.93 DRD2 (0.53) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7506072 0.92 CASP3 (0.46) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7501250 0.92 DRD2 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7501245 0.92 DRD2 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E
Bromide SCHEMBL9081927 0.91 DRD2 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E
Bromide SCHEMBL9081924 0.91 DRD2 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7508044 0.90 BRD4 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E
SCHEMBL7508040 0.90 BRD4 (0.43) DRD2DRD4HSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed