SCHEMBL7501371

SCHEMBL7501371

CCSC(=O)C(C#N)=C(C)NCC(C)C

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MMP1 P03956 1/20 0.33
MMP8 P22894 1/20 0.33
EPHX1 P07099 1/20 0.32
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501368 1.00 CYP2D6 (0.36) CYP2D6CYP2C19MMP1MMP8EPHX1
SCHEMBL7493927 0.78 MCL1 (0.32)
SCHEMBL7493932 0.78 MCL1 (0.32)
SCHEMBL7494433 0.75 ALDH1A1 (0.42) CYP2D6CYP2C19MMP1MMP8MAPT
SCHEMBL2086355 0.74 ALDH1A1 (0.36) TSHR
SCHEMBL7496095 0.73 ALDH1A1 (0.56) CYP2C19TSHR
SCHEMBL7496099 0.73 ALDH1A1 (0.56) CYP2C19TSHR
SCHEMBL5231668 0.70 TSHR (0.33) CYP2D6CYP2C19MAPTTSHR
SCHEMBL5231676 0.70 TSHR (0.33) CYP2D6CYP2C19MAPTTSHR
SCHEMBL5231682 0.70 TSHR (0.33) CYP2D6CYP2C19MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760362-B1 DIAMINOMETHYLIDENE DERIVATIVE NISSHIN SEIFUN GROUP INC (JP) 2002-08-14 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed