SCHEMBL7501744

SCHEMBL7501744

COc1ccc(CCNc2ccnc3cc(Cl)ccc23)cc1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.65
HTR1A P08908 2/20 0.64
ADRA1D P25100 2/20 0.64
ADRA1A P35348 2/20 0.64
ADRA1B P35368 2/20 0.64
HRH3 Q9Y5N1 1/20 0.64
CCR1 P32246 1/20 0.62
FERMT2 Q96AC1 4/20 0.60
CCNC P24863 1/20 0.58
CDK8 P49336 1/20 0.58
KDM4E B2RXH2 1/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
HSD17B10 Q99714 1/20 0.57
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7509385 0.91 CYP1A2 (0.65) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL7500391 0.89 CYP1A2 (0.78) CYP1A2HRH3CCR1FERMT2CCNC
SCHEMBL7513234 0.87 CCR1 (0.62) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL7501930 0.87 HTR1A (0.66) HTR1AADRA1DADRA1AADRA1BHRH3
SCHEMBL7510312 0.86 CYP1A2 (0.70) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL7505625 0.86 HTR1A (0.69) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL13496183 0.85 PKM (0.66) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL21855417 0.84 CYP1A2 (0.70) CYP1A2HRH3CCR1FERMT2CCNC
SCHEMBL31020168 0.84 CYP1A2 (0.70) CYP1A2HRH3CCR1FERMT2CCNC
SCHEMBL7503073 0.84 CCNC (0.81) CYP1A2CCR1FERMT2CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0326331-B1 Substituted quinolines and cinnolines DOW AGROSCIENCES LLC (US) 2002-04-17 EP disclosed