SCHEMBL7502452

SCHEMBL7502452

COc1ccc(C(N)=O)cc1N1CCN(Cc2cccc(-c3ccccc3)c2)CC1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.69
HTR7 P34969 2/20 0.58
POLB P06746 1/20 0.57
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
RECQL P46063 1/20 0.53
DRD2 P14416 8/20 0.51
DRD3 P35462 6/20 0.51
FAAH O00519 5/20 0.51
HTR1A P08908 3/20 0.51
UTS2R Q9UKP6 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7989214 0.99 DRD4 (0.68) DRD4HTR7POLBKMT2AKDM4E
SCHEMBL7034866 0.92 HTR7 (0.57) DRD4HTR7POLBALDH1A1LMNA
SCHEMBL7506230 0.90 DRD4 (0.56) DRD4HTR7POLBKMT2AKDM4E
SCHEMBL7498001 0.85 DRD4 (0.53) DRD4KMT2AKDM4EMEN1ALDH1A1
SCHEMBL7991732 0.82 DRD4 (1.00) DRD4HTR7POLBKMT2AKDM4E
Fumaric Acid SCHEMBL7977401 0.81 DRD4 (0.83) DRD4HTR7POLBDRD2DRD3
Maleic Acid SCHEMBL7977396 0.81 DRD4 (0.83) DRD4HTR7POLBDRD2DRD3
SCHEMBL7507348 0.79 DRD4 (0.72) DRD4HTR7POLBKDM4EALDH1A1
SCHEMBL12962319 0.78 DRD4 (0.91) DRD4HTR7POLBKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7989155 0.78 DRD4 (0.71) DRD4HTR7POLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931067-B1 D4 RECEPTOR SELECTIVITY PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2002-06-26 EP disclosed
US-6258813-B1 BIOLOGICAL RECEPTORS WITH TETRAHYDROPIPERIZINE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT (DE) 2001-07-10 US disclosed