SCHEMBL7502802

SCHEMBL7502802

COc1ccc(N)cc1OCC(C)N(C)C

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
GAA P10253 3/20 0.57
KDM4E B2RXH2 4/20 0.49
MAPT P10636 3/20 0.49
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
CYP19A1 P11511 2/20 0.41
NR4A1 P22736 1/20 0.41
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.38
HTR2A P28223 1/20 0.38
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7265202 0.83 ALDH1A1 (0.80) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL6176115 0.81 GAA (0.49) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL10187288 0.77 ALDH1A1 (0.80) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL6925643 0.76 GAA (0.46) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL7403010 0.76 SMN1; SMN2 (0.50) ALDH1A1MAPTHTTCYP19A1LMNA
SCHEMBL7404286 0.76 KDM4E (0.45) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL1130003 0.75 KDM4E (0.57) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL21663432 0.75 ALDH1A1 (0.46) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL9570228 0.74 ALDH1A1 (0.96) ALDH1A1GAAKDM4EMAPTTSHR
SCHEMBL31098523 0.74 GAA (0.82) ALDH1A1GAAKDM4EMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5801170-A Heterocyclic biphenylylamides useful as 5HT1D antagonists SMITHKLINE BEECHAM PLC (GB) 1998-09-01 US disclosed
EP-0733048-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-09-25 EP disclosed
WO-1995015954-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-06-15 WO disclosed