SCHEMBL7404286

SCHEMBL7404286

COc1ccc(N)cc1OC(C)N(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
GAA P10253 3/20 0.45
MAPT P10636 3/20 0.45
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
NR4A1 P22736 1/20 0.44
ALDH1A1 P00352 6/20 0.42
USP2 O75604 1/20 0.42
CYP19A1 P11511 2/20 0.41
LMNA P02545 1/20 0.41
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
ATM Q13315 1/20 0.36
AOC3 Q16853 1/20 0.36
IMPDH2 P12268 1/20 0.36
IMPDH1 P20839 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6902130 0.85 KDM4E (0.44) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL1010304 0.82 KDM4E (0.50) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL8687840 0.79 KDM4E (0.45) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL27939656 0.79 GAA (0.49) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL2438047 0.77 KDM4E (0.67) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL77823 0.77 KDM4E (0.67) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL29377777 0.77 KDM4E (0.67) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL4323659 0.77 KDM4E (0.49) KDM4EGAAMAPTTSHRMAPK1
SCHEMBL7502802 0.76 ALDH1A1 (0.57) KDM4EGAAMAPTTSHRMAPK1
Ammonia Solution, Strong SCHEMBL5361377 0.75 KDM4E (0.64) KDM4EGAAMAPTTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5801170-A Heterocyclic biphenylylamides useful as 5HT1D antagonists SMITHKLINE BEECHAM PLC (GB) 1998-09-01 US disclosed
EP-0733048-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-09-25 EP disclosed
WO-1995015954-A1 HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-06-15 WO disclosed