SCHEMBL7510167

SCHEMBL7510167

C1CCC(CCNC2=NCCO2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 12/20 0.53
ADRA2B P18089 12/20 0.53
ADRA2C P18825 12/20 0.53
ADRA1A P35348 4/20 0.53
CYP3A4 P08684 2/20 0.41
GMNN O75496 1/20 0.41
CYP1A2 P05177 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
OPRK1 P41145 1/20 0.41
HIF1A Q16665 1/20 0.41
NISCH Q9Y2I1 1/20 0.41
CA2 P00918 1/20 0.38
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
CHRM2 P08172 3/20 0.35
CHRM1 P11229 3/20 0.35
CHRM3 P20309 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4401199 0.78 ADRA2A (0.45) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL9558819 0.75 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL9558829 0.72 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL11710024 0.71 ADRA2A (0.73) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL11710014 0.71 ADRA2A (0.73) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL11125378 0.71
SCHEMBL1726232 0.67 SMN1; SMN2 (0.43) ADRA2AADRA2BADRA2CADRA1ACYP3A4
SCHEMBL24533674 0.66
SCHEMBL10143149 0.66
SCHEMBL11356202 0.66 ADRA2A (0.39) ADRA2AADRA2BADRA2CADRA1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1044194-A4 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS UNIV MELBOURNE (AU) 2002-01-09 EP disclosed
EP-1044194-A1 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS THE UNIVERSITY OF MELBOURNE (AU) 2000-10-18 EP disclosed
WO-1999024411-A1 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS THE UNIVERSITY OF MELBOURNE (AU) 1999-05-20 WO disclosed