SCHEMBL7511048

SCHEMBL7511048

N#Cc1ccc(N)c(OC(=O)C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 2/20 0.36
PTGDR2 Q9Y5Y4 4/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
MLYCD O95822 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TRPV4 Q9HBA0 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
PTGS2 P35354 1/20 0.34
USP30 Q70CQ3 1/20 0.34
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP2 Q9UGN5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL224235 0.76 HRH4 (0.49) TRPV4PDK2
SCHEMBL28327501 0.74 F2 (0.46) MLYCDHDAC1HDAC6PARP15PARP10
SCHEMBL7076049 0.72 ALDH1A1 (0.56) PTGDR2MRGPRX4TRPV4
Trifluoroacetic Acid SCHEMBL7511044 0.72 CXCR2 (0.41) MLYCDHDAC1HDAC6TRPV4TMPRSS4
SCHEMBL29559790 0.71 ALDH1A1 (0.57)
SCHEMBL220780 0.71 ALDH1A1 (0.57)
SCHEMBL7076047 0.71 HRH4 (0.38) PTGDR2MRGPRX4TRPV4
SCHEMBL16336032 0.70 MKNK2 (0.40) PTGDR2TRPV4
SCHEMBL15184491 0.69 SLC22A12 (0.36) TRPV4
SCHEMBL28142832 0.69 ENPP2 (0.38) NCEH1PTGDR2TRPV4PARP15PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107948-A4 AN IMPROVED SYNTHESIS OF 3-HYDROXY-4-AMINO-BENZONITRILE SMITHKLINE BEECHAM (US) 2002-01-02 EP disclosed
EP-1107948-A1 AN IMPROVED SYNTHESIS OF 3-HYDROXY-4-AMINO-BENZONITRILE Smithkline Beecham (US) 2001-06-20 EP disclosed
WO-2000012468-A1 AN IMPROVED SYNTHESIS OF 3-HYDROXY-4-AMINO-BENZONITRILE SMITHKLINE BEECHAM CORPORATION (US) 2000-03-09 WO disclosed