SCHEMBL7511491

SCHEMBL7511491

O=c1[nH]nnc2nn(Cc3ccc(Cl)cc3)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
ADORA3 P0DMS8 2/20 0.39
NOTUM Q6P988 1/20 0.38
ROCK2 O75116 1/20 0.37
PIM1 P11309 1/20 0.37
KDR P35968 1/20 0.37
GSK3B P49841 1/20 0.37
AURKB Q96GD4 1/20 0.37
PTGS2 P35354 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510532 0.88 LMNA (0.41) LMNAADORA3ROCK2GSK3BPTGS2
SCHEMBL7510407 0.87 ADORA3 (0.51) ADORA3ADORA2AADORA1CYP1A2CYP2C9
SCHEMBL7509410 0.86 TYR (0.44) ADORA3ROCK2KDRGSK3BAURKB
SCHEMBL7516038 0.80 LMNA (0.43) LMNAADORA3ROCK2PIM1GSK3B
SCHEMBL7509548 0.76 KMT2A (0.44) LMNAALDH1A1CYP2C19HTTSMN1; SMN2
SCHEMBL7515739 0.75 MKNK1 (0.43) LMNAADORA3ADORA2AADORA1ALDH1A1
SCHEMBL7514619 0.75 AR (0.42) ROCK2PIM1GSK3BAURKBALDH1A1
SCHEMBL7513782 0.72 AR (0.45) ADORA2AADORA1ALDH1A1NPSR1DAO
SCHEMBL7479263 0.65 MAPT (0.52) ADORA3ADORA2AADORA1ALDH1A1SMN1; SMN2
SCHEMBL7478026 0.63 ADORA3 (0.45) ADORA3GSK3BALDH1A1DAOPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181292-A1 PYROZOLO [3,4-D][1,2,3] TRIAZINES WITH AN ANTICONVULSIVE ACTION AND METHODS FOR PRODUCING THE SAME ARZNEIMITTELWERK DRESDEN GMBH (DE) 2002-02-27 EP claimed
WO-2000073309-A1 PYROZOLO [3,4-D][1,2,3] TRIAZINES WITH AN ANTICONVULSIVE ACTION AND METHODS FOR PRODUCING THE SAME ARZNEIMITTELWERK DRESDEN GMBH (DE) 2000-12-07 WO claimed
US-6316448-B1 Pyrazolo[3,4-d][1,2,3] troazines having anticonvulsant activity and process for their preparation ZENTARIS GMBH (DE) 2001-11-13 US disclosed