SCHEMBL7511865

SCHEMBL7511865

O=CCCc1ccccc1OCC(O)CN1CCC(Oc2ccc(Cl)cc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 6/20 0.49
DRD2 P14416 4/20 0.49
DRD3 P35462 3/20 0.49
CCR1 P32246 1/20 0.46
HRH1 P35367 1/20 0.46
CCR3 P51677 1/20 0.46
HSD17B10 Q99714 1/20 0.45
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
ADRB2 P07550 4/20 0.42
ADRB1 P08588 4/20 0.42
ADRB3 P13945 4/20 0.42
MAPT P10636 1/20 0.42
CACNA1G O43497 1/20 0.41
KCNH2 Q12809 1/20 0.41
RECQL P46063 1/20 0.41
CYP2D6 P10635 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7069082 0.94 DRD4 (0.56) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7513106 0.92 DRD4 (0.50) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7511059 0.92 DRD4 (0.50) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7512148 0.90 HRH1 (0.57) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7509383 0.89 DRD2 (0.45) DRD4DRD2DRD3CCR1HRH1
SCHEMBL28750368 0.87 DRD4 (0.49) DRD4DRD2DRD3CCR1HRH1
SCHEMBL6216294 0.86 CCR1 (0.47) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7512915 0.86 DRD4 (0.57) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7508560 0.86 DRD4 (0.57) DRD4DRD2DRD3CCR1HRH1
SCHEMBL7508179 0.85 HRH1 (0.63) DRD4DRD2DRD3CCR1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263724-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062728-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-08-30 WO disclosed