SCHEMBL7512148

SCHEMBL7512148

O=CCCc1ccccc1OCC(O)CN1CCC(Oc2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 15/20 0.57
CCR3 P51677 15/20 0.57
CCR1 P32246 2/20 0.57
DRD2 P14416 4/20 0.45
DRD4 P21917 4/20 0.45
DRD3 P35462 3/20 0.45
KCNH2 Q12809 8/20 0.44
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7508179 0.95 HRH1 (0.63) HRH1CCR3CCR1DRD2DRD4
SCHEMBL7499464 0.92 HRH1 (0.58) HRH1CCR3CCR1DRD2DRD4
SCHEMBL7511865 0.90 DRD4 (0.49) HRH1CCR3CCR1DRD2DRD4
SCHEMBL7509383 0.88 DRD2 (0.45) HRH1CCR3CCR1DRD2DRD4
SCHEMBL7511059 0.88 DRD4 (0.50) HRH1CCR3CCR1DRD2DRD4
SCHEMBL6214791 0.87 HRH1 (0.58) HRH1CCR3CCR1KCNH2
SCHEMBL7069082 0.85 DRD4 (0.56) HRH1CCR3CCR1DRD2DRD4
SCHEMBL6213285 0.84 HRH1 (0.60) HRH1CCR3CCR1DRD2DRD4
SCHEMBL7507260 0.83 CCR3 (0.54) HRH1CCR3CCR1DRD2DRD4
SCHEMBL6211818 0.82 HRH1 (0.61) HRH1CCR3CCR1KCNH2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263724-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062728-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263724-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2002-12-11 EP disclosed
EP-1263760-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062757-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-08-30 WO disclosed
WO-2001062728-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-08-30 WO disclosed