SCHEMBL7512216

SCHEMBL7512216

O=C1NCC(=O)N2Cc3cc([N+](=O)[O-])ccc3CC12

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PNMT P11086 11/20 0.47
ADRA2A P08913 7/20 0.47
ADRA2B P18089 3/20 0.47
ADRA2C P18825 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7511291 0.70 PNMT (0.41) PNMTADRA2AADRA2BADRA2C
SCHEMBL18263915 0.69 CRBN (0.43)
SCHEMBL26597131 0.68 HTR2C (0.43) PNMTADRA2A
Hydrochloric Acid SCHEMBL30643257 0.67 HTR2C (0.42) PNMTADRA2A
SCHEMBL24869941 0.66 PNMT (0.55) PNMTADRA2AADRA2BADRA2C
SCHEMBL11731134 0.66 PNMT (0.42) PNMTADRA2AADRA2BADRA2C
SCHEMBL11731123 0.66 PNMT (0.42) PNMTADRA2AADRA2BADRA2C
SCHEMBL2061424 0.66 PNMT (0.58) PNMTADRA2AADRA2BADRA2C
SCHEMBL1398082 0.65 CRBN (0.43) PNMTADRA2AADRA2BADRA2C
SCHEMBL29370265 0.65 PNMT (0.57) PNMTADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP disclosed
US-6140322-A Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase ASTRA AKTIEBOLAG (SE) 2000-10-31 US disclosed
US-5929085-A Amidine and isothiourea derivatives, compositions containing them and their use as inhibitors of nitric oxide synthase ASTRA AKTIEBOLAG (SE) 1999-07-27 US disclosed