SCHEMBL7511291

SCHEMBL7511291

O=C1COCC2Cc3ccc([N+](=O)[O-])cc3CN12

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PNMT P11086 10/20 0.41
ADRA2A P08913 7/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
NOTUM Q6P988 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7516598 0.75 ALDH1A1 (0.44) PNMTADRA2AADRA2BADRA2C
SCHEMBL21526447 0.74 DPP7 (0.41) PNMTADRA2AADRA2BADRA2C
SCHEMBL11731123 0.71 PNMT (0.42) PNMTADRA2AADRA2BADRA2C
SCHEMBL11731134 0.71 PNMT (0.42) PNMTADRA2AADRA2BADRA2C
SCHEMBL28564313 0.71 TERT (0.44)
SCHEMBL30561533 0.70 PNMT (0.43) PNMTADRA2A
SCHEMBL20704027 0.70 PNMT (0.43) PNMTADRA2A
SCHEMBL7512216 0.70 PNMT (0.47) PNMTADRA2AADRA2BADRA2C
SCHEMBL308120 0.69 ALDH1A1 (0.52) PNMTADRA2AADRA2BADRA2C
SCHEMBL22944317 0.68 HDAC6 (0.44) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP disclosed
US-6140322-A Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase ASTRA AKTIEBOLAG (SE) 2000-10-31 US disclosed
EP-0861250-A1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE Astra Aktiebolag (SE) 1998-09-02 EP disclosed
WO-1997017344-A1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRA AKTIEBOLAG (SE) 1997-05-15 WO disclosed