SCHEMBL7513003

SCHEMBL7513003

CC(=O)O[C@@H]1OCC[C@@H]1NC(=O)[C@H](CC(C)C)NC(=O)CCCN(C=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.52
CAPNS1 P04632 4/20 0.51
CTSK P43235 7/20 0.42
CTSL P07711 2/20 0.42
CTSS P25774 2/20 0.42
CTSB P07858 1/20 0.42
CASP1 P29466 4/20 0.41
CASP3 P42574 4/20 0.41
CASP7 P55210 4/20 0.41
CASP6 P55212 3/20 0.41
CASP8 Q14790 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7517808 0.92 CAPN1 (0.43) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL7515359 0.89 CAPN1 (0.56) CAPN1CAPNS1CASP1CASP3CASP7
SCHEMBL7512998 0.82 CAPN1 (0.53) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL7514161 0.81 CAPN1 (0.57) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL7511787 0.80 CAPN1 (0.44) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL3577128 0.80 CTSK (0.62) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL8406499 0.80 CTSK (0.62) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL7514109 0.80 CTSK (0.62) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL7525753 0.78 CTSK (0.61) CAPN1CAPNS1CTSKCTSLCTSS
SCHEMBL8408050 0.76 CAPN1 (0.51) CAPN1CAPNS1CASP1CASP3CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed