SCHEMBL7511787

SCHEMBL7511787

O=CN(CCCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCOC1O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 8/20 0.44
CAPNS1 P04632 3/20 0.42
CTSK P43235 3/20 0.38
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
CTSL P07711 1/20 0.38
YAP1 P46937 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515359 0.91 CAPN1 (0.56) CAPN1CAPNS1
SCHEMBL7517808 0.88 CAPN1 (0.43) CAPN1CAPNS1CTSKCTSBCTSS
SCHEMBL7513003 0.80 CAPN1 (0.52) CAPN1CAPNS1CTSKCTSBCTSS
SCHEMBL7511780 0.80 BMP1 (0.51) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL8812581 0.77 CTSK (0.60) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL8812573 0.77 CTSK (0.60) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL7514986 0.74 CAPN1 (0.52) CAPN1CAPNS1
SCHEMBL7514977 0.72 CAPN1 (0.59) CAPN1CAPNS1
SCHEMBL7516532 0.72 CTSS (0.56) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL27427437 0.72 CTSS (0.56) CAPN1CTSKCTSBCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed