SCHEMBL7513372

SCHEMBL7513372

O=[N+]([O-])c1cc2c(Cl)nc(-c3ccncc3)nc2s1.O=[N+]([O-])c1cccc(CNc2nc(-c3ccncc3)nc3sc([N+](=O)[O-])cc23)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 8/20 0.55
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
ATM Q13315 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
KCNN3 Q9UGI6 1/20 0.41
PTGS1 P23219 1/20 0.41
TBXAS1 P24557 1/20 0.41
PTGS2 P35354 1/20 0.41
PRKCI P41743 3/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5128123 0.95 PDE5A (0.60) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5128315 0.88 PDE5A (0.59) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5815431 0.87 PTGS2 (0.43) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5119410 0.85 PDE5A (0.57) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5126440 0.85 PDE5A (0.62) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5129296 0.85 PDE5A (0.59) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL7521883 0.84 KDM4E (0.53) PDE5AMEN1KMT2AMAPTATM
SCHEMBL5122225 0.84 PRKCI (0.42) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL8185259 0.83 PDE5A (0.60) PDE5AMEN1KMT2AALDH1A1POLB
SCHEMBL5129048 0.83 PRKCI (0.58) PDE5AMEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920431-A1 THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 1999-06-09 EP disclosed
WO-1998006722-A1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed