SCHEMBL7514653

SCHEMBL7514653

CC1Cc2ccc(N=C(N)c3cccs3)cc2CN1C

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 15/20 0.67
NOS1 P29475 16/20 0.53
NOS2 P35228 13/20 0.53
KCNH2 Q12809 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510902 0.86 NOS3 (0.63) NOS3NOS1NOS2KCNH2
SCHEMBL7828344 0.80 NOS3 (1.00) NOS3NOS1NOS2KCNH2
Hydrochloric Acid SCHEMBL7827939 0.79 NOS3 (0.98) NOS3NOS1NOS2
SCHEMBL7511924 0.78 NOS3 (0.63) NOS3NOS1NOS2KCNH2
SCHEMBL7513065 0.78 NOS3 (0.64) NOS3NOS1NOS2KCNH2
Hydrochloric Acid SCHEMBL7511295 0.77 NOS3 (0.61) NOS3NOS1NOS2KCNH2
SCHEMBL7510808 0.77 NOS3 (0.63) NOS3NOS1NOS2KCNH2
SCHEMBL7511533 0.76 NOS3 (0.65) NOS3NOS1NOS2KCNH2
SCHEMBL7826140 0.76 NOS3 (0.76) NOS3NOS1NOS2KCNH2
SCHEMBL7516223 0.76 NOS1 (0.64) NOS3NOS1NOS2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP disclosed
US-6140322-A Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase ASTRA AKTIEBOLAG (SE) 2000-10-31 US disclosed
US-5929085-A Amidine and isothiourea derivatives, compositions containing them and their use as inhibitors of nitric oxide synthase ASTRA AKTIEBOLAG (SE) 1999-07-27 US disclosed