SCHEMBL7516109

SCHEMBL7516109

[N-]=[N+]=CCC(=O)Oc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.44
ELANE P08246 1/20 0.40
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALOX15 P16050 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL564747 0.77 CYP19A1 (0.49) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL7520802 0.76 ALDH1A1 (0.56) TDP1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7693338 0.76 ELANE (0.47) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL9387868 0.76 CYP19A1 (0.47) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL163578 0.76 ALDH1A1 (0.50) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL6592746 0.76 CYP19A1 (0.47) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL4888627 0.74 CYP19A1 (0.46) CYP19A1ELANEPRSS1PRSS2PRSS3
Bicarbonate SCHEMBL27510048 0.74 ALDH1A1 (0.49) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL2788102 0.74 ALDH1A1 (0.49) CYP19A1ELANEPRSS1PRSS2PRSS3
SCHEMBL81292 0.73 NPSR1 (0.48) ELANEMAPTTDP1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1169328-A2 AVERMECTIN DERIVATIVES Bayer Aktiengesellschaft (DE) 2002-01-09 EP disclosed
WO-2000058328-A2 AVERMECTIN DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-10-05 WO disclosed