SCHEMBL7517595

SCHEMBL7517595

CN1CC(C(=O)N(CCCN2CCC(Cc3ccccc3)CC2)C2Cc3ccccc3C2)CC1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.51
OPRM1 P35372 4/20 0.47
ADRB2 P07550 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
ADRB1 P08588 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
DRD2 P14416 1/20 0.46
CHRM3 P20309 1/20 0.46
DRD4 P21917 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
DRD3 P35462 1/20 0.46
CCR3 P51677 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
PARP1 P09874 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455496 0.85 OPRM1 (0.58) CCR5OPRM1CCR3SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL7465772 0.83 CCR5 (0.70) CCR5OPRM1
SCHEMBL7470084 0.81 OPRM1 (0.53) CCR5OPRM1ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7470211 0.80 CCR5 (0.63) CCR5OPRM1
Hydrochloric Acid SCHEMBL7463538 0.80 CCR5 (0.56) CCR5OPRM1
Hydrochloric Acid SCHEMBL7453187 0.80 CCR5 (0.63) CCR5OPRM1
Hydrochloric Acid SCHEMBL7454310 0.80 CCR5 (0.55) CCR5OPRM1
Hydrochloric Acid SCHEMBL7464027 0.79 CCR5 (0.59) CCR5OPRM1CCR3
SCHEMBL7465426 0.79 SLC6A2 (0.49) CCR5OPRM1
SCHEMBL3038736 0.79 CCR5 (0.62) CCR5OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180513-A1 CYCLIC AMIDE COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-20 EP disclosed