SCHEMBL7517826

SCHEMBL7517826

Cn1nc(-c2cc(C(=O)O)c(Cl)cc2F)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.40
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GAA P10253 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
TTR P02766 1/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NTRK1 P04629 5/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27519042 0.82 ALDH1A1 (0.39) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL7521846 0.80 ALDH1A1 (0.37) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL30130331 0.80 ALDH1A1 (0.37) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL4067277 0.78 NTRK1 (0.37) MAPTMEN1KMT2ANTRK1
SCHEMBL1700760 0.77 CYP1A2 (0.37) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL8333887 0.77 ALDH1A1 (0.43) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL27989452 0.76 ALDH1A1 (0.47) ALDH1A1PKMSMN1; SMN2GAAL3MBTL1
SCHEMBL8546587 0.76 RORC (0.36) ALDH1A1L3MBTL1NTRK1
SCHEMBL27500378 0.75 LMNA (0.47) ALDH1A1PKMMAPTSMN1; SMN2NPSR1
SCHEMBL27463655 0.75 ALDH1A1 (0.37) ALDH1A1PKMMAPTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772598-B1 PREPARATION OF HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS MONSANTO TECHNOLOGY LLC (US) 2002-02-06 EP disclosed
US-6121458-A ACYLATION, HALOGENATION, ALKYLATION, CATALYTIC OXIDATION, AND ESTERIFICATION; CYCLIZATION AND CONDENSATION WITH HYDRAZINE MONSANTO COMPANY (US) 2000-09-19 US disclosed
US-5986104-A ESTERIFICATION OF ACID COMPOUNDS FORMED BY OXIDATION OF METHYL GROUPS TO FORM HERBICIDES MONSANTO COMPANY (US) 1999-11-16 US disclosed
US-5973164-A Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity MONSANTO COMPANY (US) 1999-10-26 US disclosed
US-5969153-A CONDENSING A PHENYL DIKETONE WITH HYDRAZINE IN SOLVENT, THEN ALKYLATION MONSANTO COMPANY (US) 1999-10-19 US disclosed
EP-0923520-A2 PREPARATION OF SUBSTITUTED 3-ARYL-5-HALOALKYL-PYRAZOLES HAVING HERBICIDAL ACTIVITY MONSANTO COMPANY (US) 1999-06-23 EP disclosed
WO-1997048668-A2 PREPARATION OF SUBSTITUTED 3-ARYL-5-HALOALKYL-PYRAZOLES HAVING HERBICIDAL ACTIVITY MONSANTO COMPANY (US) 1997-12-24 WO disclosed
EP-0772598-A1 HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS AND SYNTHESIS THEREOF MONSANTO COMPANY (US) 1997-05-14 EP disclosed
US-5587485-A CATALYTIC OXIDATION OF THE CORRESPONDING ALKYL SUBSTITUTED BENZENE COMPOUND MONSANTO COMPANY (US) 1996-12-24 US disclosed
WO-1996002515-A1 HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS AND SYNTHESIS THEREOF MONSANTO COMPANY (US) 1996-02-01 WO disclosed