SCHEMBL7519979

SCHEMBL7519979

O=C(O)OC1Cc2c([nH]c3ccccc23)C(c2ccccc2)N1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.67
TSHR P16473 2/20 0.67
MAPK1 P28482 1/20 0.67
CCKBR P32239 2/20 0.54
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
CYP2C19 P33261 2/20 0.52
ALOX12 P18054 1/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HTT P42858 2/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
HTR7 P34969 1/20 0.49
CYP3A4 P08684 1/20 0.49
HSD17B10 Q99714 2/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7522074 0.90 SSTR3 (0.58) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL7525817 0.85 KDM4E (0.62) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL4787100 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL28478851 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL17760630 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL764194 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL29630317 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL3481444 0.80 CYP2D6 (1.00) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL7523636 0.80 CYP2D6 (0.53) CYP2D6TSHRMAPK1CCKBRMEN1
SCHEMBL7520532 0.79 MEN1 (0.50) CYP2D6TSHRMAPK1CCKBRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891187-B1 USE OF DERIVATIVES OF TETRAHYDRO-BETA-CARBOLINES AS ANTIMETASTATIC AGENTS HOFFMANN LA ROCHE (CH) 2002-01-30 EP claimed