SCHEMBL7520262

SCHEMBL7520262

CC(=O)NC(C(=O)NCc1ccc(F)cc1)c1ccco1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.48
ALDH1A1 P00352 4/20 0.48
LMNA P02545 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 2/20 0.44
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8837220 1.00 CCR2 (0.48) CCR2ALDH1A1LMNAMEN1KMT2A
SCHEMBL8837195 0.89 NPSR1 (0.55) CCR2ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL6813763 0.88 CA12 (0.54) CCR2ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1710436 0.87 CCR2 (0.48) CCR2ALDH1A1MEN1KMT2AHPGD
SCHEMBL8837111 0.87 CCR2 (0.56) CCR2SMN1; SMN2KDM4ENPSR1
SCHEMBL9712175 0.87 CCR2 (0.56) CCR2SMN1; SMN2KDM4ENPSR1
SCHEMBL8837129 0.85 ALDH1A1 (0.48) CCR2ALDH1A1LMNASMN1; SMN2
SCHEMBL8837177 0.84 CCR2 (0.43) CCR2ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7521866 0.83 CCR2 (0.43) CCR2ALDH1A1LMNAHPGDKDM4E
SCHEMBL7522219 0.82 CCR2 (0.43) CCR2ALDH1A1LMNAKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400440-B1 Amino acid derivative anticonvulsant RES CORP TECHNOLOGIES INC (US) 2002-03-13 EP claimed
US-5378729-A Diamide derivatives RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1995-01-03 US claimed
WO-1990015069-A2 AMINO ACID DERIVATIVE ANTICONVULSANT RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-12-13 WO claimed
EP-0400440-A1 Amino acid derivative anticonvulsant RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-12-05 EP claimed
EP-1218370-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS Aventis Pharma S.A. (FR) 2002-07-03 EP disclosed
EP-0400440-B1 Amino acid derivative anticonvulsant RES CORP TECHNOLOGIES INC (US) 2002-03-13 EP disclosed
WO-2001025227-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2001-04-12 WO disclosed
US-5654301-A Lacosamide FDA Orange book listed patent RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1997-08-05 US disclosed
US-5378729-A Diamide derivatives RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1995-01-03 US disclosed
EP-0400440-A1 Amino acid derivative anticonvulsant RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-12-05 EP disclosed