SCHEMBL7521149

SCHEMBL7521149

CCc1cccc([SiH2]CSc2ccc(O)c(C(C)(C)C)c2)c1CC

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.34
HSP90AB1 P08238 2/20 0.34
ALDH1A1 P00352 2/20 0.34
NR1I2 O75469 1/20 0.34
LMNA P02545 1/20 0.34
CYP2C9 P11712 1/20 0.34
MIF P14174 1/20 0.34
TYR P14679 1/20 0.34
ALOX15 P16050 1/20 0.34
HTT P42858 1/20 0.34
NFE2L2 Q16236 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
GAA P10253 1/20 0.30
XBP1 P17861 1/20 0.30
ATM Q13315 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7516049 0.86 NR1I2 (0.33) HSP90AA1HSP90AB1ALDH1A1NR1I2LMNA
SCHEMBL7519331 0.84 NPSR1 (0.32) HSP90AA1HSP90AB1ALDH1A1NR1I2LMNA
SCHEMBL7521936 0.84 ALDH1A1 (0.35) ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL7526671 0.83 GABRA1 (0.35) ALDH1A1NR1I2LMNACYP2C9MIF
SCHEMBL7526427 0.81 ALDH1A1 (0.37) HSP90AA1HSP90AB1ALDH1A1NR1I2LMNA
SCHEMBL7525374 0.80 ALDH1A1 (0.36) HSP90AA1HSP90AB1ALDH1A1NR1I2LMNA
SCHEMBL7521636 0.76 NR1I2 (0.33) ALDH1A1NR1I2LMNACYP2C9MIF
SCHEMBL8442028 0.74 GABRA1 (0.36) HSP90AA1HSP90AB1GABRA1GABRB2L3MBTL1
SCHEMBL7525678 0.72 GABRA1 (0.33) GABRA1GABRB2
SCHEMBL27515458 0.71 ESR1 (0.34) HSP90AA1HSP90AB1HSD17B10GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed