SCHEMBL7521287

SCHEMBL7521287

CCCCc1nn2ccccc2c1Cc1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.40
MMP12 P39900 1/20 0.40
HDAC1 Q13547 3/20 0.39
AGTR1 P30556 4/20 0.37
PPARG P37231 3/20 0.37
KCNH2 Q12809 1/20 0.37
NPC1 O15118 1/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADCY10 Q96PN6 1/20 0.36
EGFR P00533 1/20 0.34
AGTR2 P50052 1/20 0.34
CXCR3 P49682 1/20 0.34
CNR2 P34972 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878871 0.83 MMP3 (0.36) MMP3MMP12HDAC1AGTR1PPARG
SCHEMBL7518256 0.79 NPC1 (0.36) NPC1NFKB1MAPK1RAB9ANFKB2
SCHEMBL7510620 0.78 AGTR1 (0.61) AGTR1PPARGAGTR2
SCHEMBL7508623 0.77 RARB (0.40) AGTR1AGTR2
SCHEMBL7510644 0.76 AGTR1 (0.43) AGTR1PPARGAGTR2
SCHEMBL7507671 0.76 EGFR (0.45) HDAC1AGTR1PPARGNPC1RAB9A
SCHEMBL8878903 0.74 AR (0.38) SMN1; SMN2
SCHEMBL20341902 0.73 TLR7 (0.41) EGFR
Ammonia Solution, Strong SCHEMBL6629978 0.72 HDAC1 (0.41) HDAC1AGTR1PPARGKCNH2SMN1; SMN2
SCHEMBL7510474 0.72 EGFR (0.40) HDAC1AGTR1KCNH2L3MBTL1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556080-B1 Bicyclic pyridine derivatives, process for their preparation, intermediates, their use as medicaments and pharmaceutical compositions containing them AVENTIS PHARMA SA (FR) 2002-05-08 EP disclosed
US-5691347-A ANGIOTENSIN II INHIBITORS AND VASOCONSTRICTION ROUSSEL UCLAF (FR) 1997-11-25 US disclosed
US-5650414-A PYRAZOLOPYRIDINES OR IMIDAZOLOPYRIDINES ROUSSEL UCLAF (FR) 1997-07-22 US disclosed
EP-0556080-A1 Bicyclic pyridine derivatives, process for their preparation, intermediates, their use as medicaments and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1993-08-18 EP disclosed