SCHEMBL7521996

SCHEMBL7521996

CCCC(=O)Oc1c(C(C)(C)C)cc(OC[Si](C)(C)c2ccc(C(F)(F)F)cc2)cc1C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 10/20 0.38
L3MBTL1 Q9Y468 2/20 0.32
GAA P10253 2/20 0.32
XBP1 P17861 1/20 0.32
ATM Q13315 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GSK3B P49841 2/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
SQLE Q14534 1/20 0.31
MAOB P27338 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7526551 0.88 VCAM1 (0.41) VCAM1SQLE
SCHEMBL8839727 0.87 BACE1 (0.38) VCAM1CYP1A1CYP1B1PPARDPPARA
SCHEMBL7524217 0.86 VCAM1 (0.37) VCAM1L3MBTL1GAAXBP1ATM
SCHEMBL6248869 0.81 VCAM1 (0.45) VCAM1ATM
SCHEMBL7523462 0.79 VCAM1 (0.52) VCAM1NPSR1SQLE
SCHEMBL7515902 0.79 CA2 (0.41) GAAATMNPSR1SQLEALDH1A1
SCHEMBL7524096 0.79 VCAM1 (0.38) VCAM1SQLEKMT2A
SCHEMBL7523688 0.77 VCAM1 (0.35) VCAM1L3MBTL1GAAXBP1ATM
SCHEMBL7518758 0.77 VCAM1 (0.47) VCAM1
SCHEMBL6261716 0.76 VCAM1 (0.36) VCAM1PPARDPPARAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed