SCHEMBL8839727

SCHEMBL8839727

CC(=O)Oc1c(C(C)(C)C)cc(OC[Si](C)(C)c2ccc(C(F)(F)F)cc2)cc1C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C19 P33261 2/20 0.37
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAOB P27338 2/20 0.36
SRD5A2 P31213 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
PPARA Q07869 3/20 0.33
PPARD Q03181 2/20 0.33
PPARG P37231 1/20 0.33
P2RY1 P47900 1/20 0.32
VCAM1 P19320 2/20 0.32
MAPK14 Q16539 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
STAT3 P40763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7523672 0.87 BACE1 (0.39) BACE1VCAM1
SCHEMBL7521996 0.87 VCAM1 (0.38) ALDH1A1KDM4EMAOBCYP1A1CYP1B1
SCHEMBL7520303 0.86 VCAM1 (0.33) ALDH1A1VCAM1
SCHEMBL7526592 0.85 MEN1 (0.32) ALDH1A1CYP2C19HPGDVCAM1CYP1A2
SCHEMBL7515902 0.83 CA2 (0.41) ALDH1A1USP2CYP1A2
SCHEMBL8517276 0.80 ADORA3 (0.35) BACE1ALDH1A1KDM4EHPGD
SCHEMBL6261716 0.80 VCAM1 (0.36) BACE1ALDH1A1CYP2C19KDM4EUSP2
SCHEMBL8839500 0.78 BACE1 (0.41) BACE1ALDH1A1CYP2C19KDM4EUSP2
SCHEMBL6248869 0.76 VCAM1 (0.45) VCAM1
SCHEMBL7524096 0.75 VCAM1 (0.38) VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed