SCHEMBL7522573

SCHEMBL7522573

COc1cc(CC(=O)ON2C(=O)CCC2=O)ccc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
ALDH1A1 P00352 1/20 0.58
GAA P10253 1/20 0.58
NFKB1 P19838 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
ALOX5 P09917 1/20 0.48
OR51E2 Q9H255 1/20 0.48
SHBG P04278 1/20 0.47
TAAR1 Q96RJ0 2/20 0.47
MAPK1 P28482 1/20 0.47
FOS P01100 1/20 0.46
TTR P02766 1/20 0.46
JUN P05412 1/20 0.46
NR3C1 P04150 1/20 0.46
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
LMNA P02545 1/20 0.46
GLA P06280 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384707 0.89 HTT (0.51) ALDH1A1GAALMNAGLANPC1
SCHEMBL7525396 0.88 ALOX5 (0.58) TSHRALDH1A1GAANFKB1TDP1
SCHEMBL9561266 0.82 GAA (0.48) TSHRALDH1A1GAANFKB1TDP1
SCHEMBL4545404 0.81 CA2 (0.54) TSHRALDH1A1GAAHSD17B2
SCHEMBL31225941 0.81 CA2 (0.54) TSHRALDH1A1GAAHSD17B2
SCHEMBL30128009 0.79 GAA (0.73) TSHRALDH1A1GAANFKB1TDP1
SCHEMBL9040078 0.79 TSHR (0.73) TSHRALDH1A1GAANFKB1TDP1
SCHEMBL1751797 0.79 GAA (0.73) TSHRALDH1A1GAANFKB1TDP1
SCHEMBL7521195 0.79 MAPK1 (0.42) ALDH1A1GAAMAPK1LMNAGLA
SCHEMBL499428 0.79 KMT2A (0.46) TSHRALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900781-B1 Phenolic acid amides of hydroxy substituted benzylamines HAARMANN & REIMER GMBH (DE) 2002-03-20 EP claimed
US-6117365-A N-(3,4-DIHYDROXYBENZYL)-3,5-DIMETHOXY-4-HYDROXY-E-CINNAMIDE, FOR EXAMPLE; USE AS ANTIOXIDANTS OR AS FREE-RADICAL SCAVENGERS, IN PARTICULAR IN THE COSMETIC OR DERMATOLOGICAL FIELDS, AND IN FOODS HAARMANN & REIMER GMBH (DE) 2000-09-12 US claimed
US-6117365-A N-(3,4-DIHYDROXYBENZYL)-3,5-DIMETHOXY-4-HYDROXY-E-CINNAMIDE, FOR EXAMPLE; USE AS ANTIOXIDANTS OR AS FREE-RADICAL SCAVENGERS, IN PARTICULAR IN THE COSMETIC OR DERMATOLOGICAL FIELDS, AND IN FOODS HAARMANN & REIMER GMBH (DE) 2000-09-12 US disclosed