SCHEMBL7523258

SCHEMBL7523258

N#Cc1ccc(CCCl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.54
CYP2A6 P11509 2/20 0.54
KCNJ1 P48048 1/20 0.53
KCNH2 Q12809 1/20 0.53
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP19A1 P11511 5/20 0.48
DAO P14920 2/20 0.47
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
IDO1 P14902 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CA12 O43570 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1004267 0.85 LOXL2 (0.64) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL31231842 0.85 TSHR (0.58) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL10569888 0.80 TSHR (0.68) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL9640908 0.80 TSHR (0.62) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL200142 0.80 LOXL2 (0.58) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL9860834 0.79 GFER (0.42) CYP2A6MAOAMAOBALDH1A1CA2
SCHEMBL10452241 0.78 LOXL2 (0.56) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL16582463 0.78 TSHR (0.71) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL16582531 0.78 TSHR (0.71) LOXL2CYP2A6KCNJ1KCNH2TSHR
SCHEMBL10569117 0.78 TSHR (0.71) LOXL2CYP2A6KCNJ1KCNH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109232175-A A kind of preparation method of chloroethyl substituted aromatic compound 四川理工学院 2019-01-18 CN disclosed
EP-0912586-B1 FUNCTIONALIZED FERROCENYLDIPHOSPHINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE SYNGENTA PARTICIPATIONS AG (CH) 2002-01-16 EP disclosed
US-6169192-B1 LIGANDS FOR TRANSITION METAL COMPLEXES SUITABLE FOR ENANTIOSELECTIVE HYDROGENATION OF ORGANIC DOUBLE OR TRIPLE BONDS NOVARTIS AG (CH) 2001-01-02 US disclosed
EP-0912586-A1 FUNCTIONALIZED FERROCENYLDIPHOSPHINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE Novartis AG (CH) 1999-05-06 EP disclosed
WO-1998001457-A1 FUNCTIONALIZED FERROCENYLDIPHOSPHINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE NOVARTIS AG (CH) 1998-01-15 WO disclosed