SCHEMBL7525271

SCHEMBL7525271

O=C(O)CC(C=C(F)F)c1cc(Cl)nc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.33
S1PR2 O95136 1/20 0.33
GABBR2 O75899 3/20 0.31
GABBR1 Q9UBS5 3/20 0.31
LMNA P02545 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP3A4 P08684 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
NFKB1 P19838 1/20 0.31
DRD3 P35462 1/20 0.31
BLM P54132 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
MEN1 O00255 1/20 0.31
THRB P10828 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
CTSA P10619 3/20 0.30
KEAP1 Q14145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7526351 0.86 FFAR1 (0.33) FFAR1S1PR2GABBR2GABBR1LMNA
SCHEMBL7522866 0.84 S1PR2 (0.36) FFAR1S1PR2GABBR2GABBR1LMNA
SCHEMBL7523155 0.71 FFAR1 (0.44) FFAR1LMNACYP2C19TSHRKMT2A
SCHEMBL7523172 0.69 CTSA (0.42) MEN1KMT2ACTSA
SCHEMBL7528570 0.66 KDM4E (0.40) KMT2ACTSA
SCHEMBL7524734 0.66 FFAR1 (0.45) FFAR1KMT2ACTSA
SCHEMBL7522581 0.62 ALDH1A1 (0.43) FFAR1LMNAKMO
SCHEMBL7526475 0.62 FFAR1 (0.39) FFAR1GABBR2GABBR1LMNACYP2C9
SCHEMBL7522086 0.61 FFAR1 (0.43) FFAR1GABBR2GABBR1LMNACYP2C9
SCHEMBL7524496 0.61 GABBR2 (0.46) FFAR1GABBR2GABBR1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181267-A1 HALOGEN COMPOUNDS Bayer Aktiengesellschaft (DE) 2002-02-27 EP disclosed
WO-2000071500-A1 HALOGEN COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2000-11-30 WO disclosed