SCHEMBL7525520

SCHEMBL7525520

CC(C)c1cc(CC[Si](C)(C)c2ccccc2)c(C(C)C)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.39
HSP90AA1 P07900 6/20 0.38
HSP90AB1 P08238 4/20 0.36
GABRA1 P14867 2/20 0.36
GABRB2 P47870 1/20 0.36
MAPT P10636 4/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2D6 P10635 3/20 0.35
LMNA P02545 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
ALOX15 P16050 2/20 0.35
CYP2C19 P33261 2/20 0.35
HIF1A Q16665 2/20 0.35
TP53 P04637 1/20 0.35
PAX8 Q06710 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376866 0.86 HSP90AA1 (0.32) TRPV1HSP90AA1HSP90AB1
SCHEMBL7516559 0.80 CYP1A2 (0.39) TRPV1HSP90AA1HSP90AB1GABRA1GABRB2
SCHEMBL5692015 0.77 GABRA1 (0.49) TRPV1GABRA1GABRB2MAPTCYP1A2
SCHEMBL7520561 0.73 HSP90AA1 (0.37) TRPV1HSP90AA1HSP90AB1GABRA1GABRB2
SCHEMBL7522614 0.73 GABRA1 (0.40) HSP90AA1HSP90AB1GABRA1GABRB2MAPT
SCHEMBL7519181 0.72 NPSR1 (0.37) TRPV1MAPTCYP1A2CYP2D6LMNA
SCHEMBL7526680 0.71 ESR1 (0.39) MAPTCYP1A2CYP2D6LMNANPSR1
SCHEMBL7521584 0.69 ALOX15 (0.43) MAPTCYP1A2CYP2D6LMNACYP3A4
SCHEMBL7521666 0.69 TYR (0.44) MAPTLMNANPSR1CYP3A4ALOX15
SCHEMBL5693094 0.69 GABRA1 (0.45) HSP90AA1HSP90AB1GABRA1GABRB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed