SCHEMBL7526568

SCHEMBL7526568

CSc1nc(C)cc(-c2ccccc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
PKM P14618 2/20 0.56
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
HTT P42858 1/20 0.54
MAPT P10636 4/20 0.54
LMNA P02545 2/20 0.52
TP53 P04637 1/20 0.52
THRB P10828 1/20 0.52
VCP P55072 2/20 0.52
ADORA1 P30542 3/20 0.51
ADORA2A P29274 2/20 0.51
HSD17B10 Q99714 3/20 0.49
KDM4E B2RXH2 3/20 0.49
RAB9A P51151 3/20 0.49
HPGD P15428 2/20 0.49
NPC1 O15118 2/20 0.49
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13133556 0.88 MAPT (0.58) ALDH1A1MEN1KMT2AHTTMAPT
SCHEMBL5593111 0.81 MAPT (0.57) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL13111264 0.81 VCP (0.59) ALDH1A1PKMMEN1KMT2AHTT
SCHEMBL29502715 0.80 ADORA2A (0.59) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL5593348 0.80 MAPT (0.51) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7525473 0.80 MAPT (0.51) ALDH1A1PKMMEN1KMT2AHTT
SCHEMBL7521036 0.80 KDM4E (0.56) ALDH1A1MEN1KMT2AHTTMAPT
SCHEMBL1445103 0.80 MAPT (0.51) ALDH1A1PKMMEN1KMT2AHTT
SCHEMBL14267870 0.80 ADORA2A (0.59) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL3410200 0.80 ALDH1A1 (0.51) ALDH1A1PKMMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8476225-B2 Antiviral compounds GILEAD SCIENCES, INC. (US) 2013-07-02 US disclosed
EP-1181281-A2 NOVEL CARBOXYLIC ACID DERIVATIVES COMPRISING ARYL-SUBSTITUTED NITROGEN HETEROCYCLES, THEIR PRODUCTION AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000073276-A2 CARBOXYLIC ACID DERIVATIVES COMPRISING ARYL-SUBSTITUTED NITROGEN HETEROCYCLES, THEIR PRODUCTION AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2000-12-07 WO disclosed