SCHEMBL7527079

SCHEMBL7527079

COc1ccc2c3c(ccc2c1)-c1cc(OC)c(F)cc1C3c1ccc(OCCN(C)C)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.42
ESR2 Q92731 2/20 0.42
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.38
MAOB P27338 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
BRAF P15056 1/20 0.34
DPP4 P27487 2/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HCRTR1 O43613 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531367 0.83 ESR1 (0.44) ESR1ESR2KDM4EALDH1A1DPP4
SCHEMBL7530398 0.83 ESR1 (0.64) ESR1ESR2
SCHEMBL7528465 0.83 ESR1 (0.52) ESR1ESR2KDRFLT3
SCHEMBL7527453 0.83 ESR1 (0.43) ESR1ESR2KDRTDP1
SCHEMBL8965880 0.81 MEN1 (0.46) ESR1ESR2KDRFLT3MAOB
SCHEMBL7528919 0.80 ESR1 (0.41) ESR1ESR2KDR
SCHEMBL7138825 0.76 ESR1 (0.39) ESR1ESR2KDRMAOB
SCHEMBL8609168 0.75 ESR1 (0.68) ESR1ESR2FLT3
SCHEMBL7535540 0.75 ESR1 (0.47) ESR1ESR2KDM4EALDH1A1
SCHEMBL7526145 0.74 ESR1 (0.59) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832881-B1 Benzofluorene compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2002-04-03 EP disclosed
EP-0832881-A2 Benzofluorene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed