SCHEMBL7528005

SCHEMBL7528005

CCc1cc2c(cc1OC)-c1ccc3ccccc3c1C2c1ccc(O)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
GAA P10253 3/20 0.40
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
BACE1 P56817 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
RXRA P19793 1/20 0.35
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530844 0.89 KMT2A (0.40) MEN1KMT2AGAAESR1ESR2
SCHEMBL7533104 0.88 ESR1 (0.45) MEN1KMT2AESR1ESR2KDM4E
SCHEMBL7528055 0.86 MEN1 (0.40) MEN1KMT2AGAAESR1ESR2
SCHEMBL7529347 0.85 CSNK2A2 (0.38) MEN1KMT2AGAAESR1ESR2
SCHEMBL7526863 0.85 ESR1 (0.38) MEN1KMT2AGAAESR1ESR2
SCHEMBL8966375 0.80 ESR1 (0.46) MEN1KMT2AGAAESR1ESR2
SCHEMBL7525891 0.79 ESR1 (0.59) ESR1ESR2
SCHEMBL7535540 0.76 ESR1 (0.47) MEN1KMT2AGAAESR1ESR2
SCHEMBL7532969 0.76 MEN1 (0.40) MEN1KMT2AGAAESR1ESR2
SCHEMBL8966115 0.74 ESR1 (0.39) MEN1KMT2AGAAESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832881-B1 Benzofluorene compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2002-04-03 EP disclosed
EP-0832881-A2 Benzofluorene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed