SCHEMBL7526863

SCHEMBL7526863

COc1cc2c(cc1F)C(c1ccc(O)cc1)c1c-2ccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
GAA P10253 3/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RXRA P19793 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
DRD5 P21918 2/20 0.36
ABCG2 Q9UNQ0 2/20 0.36
ABCC1 P33527 1/20 0.35
ACHE P22303 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530844 0.91 KMT2A (0.40) ESR1ESR2MEN1KMT2AGAA
SCHEMBL7528055 0.88 MEN1 (0.40) ESR1ESR2MEN1KMT2AGAA
SCHEMBL7531367 0.87 ESR1 (0.44) ESR1ESR2KDM4EALDH1A1CYP19A1
SCHEMBL7529347 0.87 CSNK2A2 (0.38) ESR1ESR2MEN1KMT2AGAA
SCHEMBL7528005 0.85 MEN1 (0.42) ESR1ESR2MEN1KMT2AGAA
SCHEMBL8966375 0.81 ESR1 (0.46) ESR1ESR2MEN1KMT2AGAA
SCHEMBL7527912 0.81 ESR1 (0.46) ESR1ESR2MEN1KMT2AKDM4E
SCHEMBL7526145 0.78 ESR1 (0.59) ESR1ESR2
SCHEMBL7535540 0.77 ESR1 (0.47) ESR1ESR2MEN1KMT2AGAA
SCHEMBL7532969 0.77 MEN1 (0.40) ESR1ESR2MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832881-B1 Benzofluorene compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2002-04-03 EP disclosed
EP-0832881-A2 Benzofluorene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed