SCHEMBL7528332

SCHEMBL7528332

Cn1cncc1-c1ccc2ccn(C)c2c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
GSK3B P49841 12/20 0.43
DYRK1A Q13627 12/20 0.43
WNT1 P04628 3/20 0.43
LRRK2 Q5S007 1/20 0.43
HPGDS O60760 1/20 0.43
CYP2A6 P11509 1/20 0.42
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
CLK2 P49760 1/20 0.41
CLK3 P49761 1/20 0.41
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22874232 0.83 IDO1 (0.59) IDO1GSK3BDYRK1AWNT1HPGDS
SCHEMBL7988012 0.77 CYP2A6 (0.45) CYP2A6
SCHEMBL4515256 0.77 IDO1 (0.57) IDO1GSK3BDYRK1AWNT1HPGDS
SCHEMBL7533347 0.76 QPCT (0.39) IDO1GSK3BDYRK1AWNT1LRRK2
SCHEMBL18029231 0.75 HTR6 (0.60) CYP2A6
SCHEMBL7524692 0.74 PIK3CD (0.47) CYP2A6
SCHEMBL17559204 0.72 FGFR1 (0.51) IDO1GSK3BDYRK1AMMP2MMP13
SCHEMBL21241353 0.72 CYP2A6 (0.41) LRRK2CYP2A6
SCHEMBL17384770 0.71 LRRK2 (0.55) GSK3BDYRK1AWNT1LRRK2
SCHEMBL20916196 0.71 GSK3B (0.55) GSK3BDYRK1AWNT1CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1193027-C Substituted pyrroles HOFFMANN LA ROCHE (CH) 2005-03-16 CN disclosed
CN-1411457-A Substituted pyrroles HOFFMANN LA ROCHE (CH) 2003-04-16 CN disclosed
EP-1242409-A2 SUBSTITUTED BISINDOLYLMALEIMIDES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-25 EP disclosed
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2001046178-A2 SUBSTITUIERTE BISINDOLYMALEIMIDE F. HOFFMANN-LA ROCHE AG (CH) 2001-06-28 WO disclosed