SCHEMBL7528581

SCHEMBL7528581

COc1cc(OC)c2c(c1)-c1ccc3ccccc3c1C2c1ccc(OCCC2CCCN2C)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.41
ESR2 Q92731 2/20 0.41
CHRM3 P20309 2/20 0.41
FAAH O00519 4/20 0.40
ACP1 P24666 1/20 0.40
CHRNB4 P30926 3/20 0.39
CHRNA3 P32297 3/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB3 Q05901 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ESRRG P62508 6/20 0.39
ESRRB O95718 2/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7529608 0.92 ESR1 (0.43) ESR1ESR2CHRM3CHRNB4CHRNA3
SCHEMBL7531753 0.87 ESR1 (0.46) ESR1ESR2CHRM3FAAHACP1
SCHEMBL7532152 0.86 ESR1 (0.56) ESR1ESR2HRH3KCNH2
SCHEMBL7535261 0.85 ESR1 (0.57) ESR1ESR2HRH3KCNH2
SCHEMBL7529441 0.81 ESR1 (0.49) ESR1ESR2CHRM3CHRNB4CHRNA3
SCHEMBL7525151 0.80 ESR1 (0.58) ESR1ESR2CHRM3CHRNB4CHRNA3
SCHEMBL7144464 0.78 CHRM3 (0.39) ESR1CHRM3CHRNB4CHRNA3ESRRG
SCHEMBL7145058 0.77 EBP (0.40) ESR1ESR2CHRM3CHRNB4CHRNA3
SCHEMBL7527322 0.77 ESR1 (0.61) ESR1ESR2
SCHEMBL7532969 0.75 MEN1 (0.40) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832881-B1 Benzofluorene compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2002-04-03 EP disclosed
EP-0832881-A2 Benzofluorene compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed