SCHEMBL7528716

SCHEMBL7528716

C=CC[CH]c1nc2ccccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
NPC1 O15118 9/20 0.53
RAB9A P51151 9/20 0.53
MEN1 O00255 7/20 0.53
KMT2A Q03164 7/20 0.53
KDM4E B2RXH2 7/20 0.53
SMN1; SMN2 Q16637 6/20 0.53
HPGD P15428 5/20 0.53
PKM P14618 4/20 0.53
HSP90AA1 P07900 1/20 0.53
MAPT P10636 5/20 0.47
GAA P10253 5/20 0.47
LMNA P02545 4/20 0.47
HTT P42858 3/20 0.47
TP53 P04637 2/20 0.47
GLA P06280 2/20 0.47
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
RECQL P46063 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6717024 0.81 DDAH1 (0.56) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL1568280 0.81 ALDH1A1 (0.59) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL854115 0.78 ALDH1A1 (0.56) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL7408425 0.77 NPC1 (0.51) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL5627161 0.77 RAB9A (0.56) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL1086985 0.77 ALDH1A1 (0.81) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL1086983 0.77 ALDH1A1 (0.81) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL19119423 0.77 ALDH1A1 (0.63) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL29539476 0.77 ALDH1A1 (0.81) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL18628734 0.75 ALDH1A1 (0.49) ALDH1A1NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465889-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY GENZYME CORP (US) 2017-03-22 EP claimed
EP-1465889-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY GENZYME CORP (US) 2017-03-22 EP disclosed
EP-0871619-B1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMA (US) 2002-11-06 EP disclosed
US-6458959-B1 VIRICIDES AND ENZYME INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-10-01 US disclosed
US-6348477-B1 SUBSTITUTED PHENYL THIAZOLE DERIVATIVES AS VIRICIDES BOEHRINGER INGELHEIM(CANADA) LTD. (CA) 2002-02-19 US disclosed
US-6057451-A AMINOTHIAZOLE DERIVATIVES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-05-02 US disclosed
EP-0871619-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1998-10-21 EP disclosed
WO-1997024343-A1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-07-10 WO disclosed